SCHEMBL28320408

SCHEMBL28320408

COc1ccccc1C(O)CNC(C)(C)C

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.64
ADRB1 P08588 3/20 0.64
CYP2D6 P10635 2/20 0.64
HIF1A Q16665 2/20 0.64
NFKB1 P19838 1/20 0.64
BLM P54132 1/20 0.62
MAPT P10636 1/20 0.48
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
MAOA P21397 1/20 0.46
HTR2B P41595 1/20 0.46
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
TSHR P16473 1/20 0.44
CASP7 P55210 1/20 0.44
KMT2A Q03164 1/20 0.44
ADRB3 P13945 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11098461 0.81 ADRB2 (0.68) ADRB2ADRB1CYP2D6HIF1ANFKB1
SCHEMBL13188558 0.81 SLC6A2 (0.52) ADRB2ADRB1CYP2D6ADRA2AADRA2B
Hydrochloric Acid SCHEMBL10877628 0.80 BLM (0.55) ADRB2ADRB1CYP2D6HIF1ANFKB1
SCHEMBL2294795 0.79 ADRB2 (0.51) ADRB2ADRB1CYP2D6HIF1ANFKB1
SCHEMBL11433167 0.79 CASR (0.69) ADRB2ADRB1CYP2D6ADRB3
SCHEMBL2294900 0.79 ADRB2 (0.51) ADRB2ADRB1CYP2D6HIF1ANFKB1
Hydrochloric Acid SCHEMBL11285463 0.79 BLM (0.47) ADRB2ADRB1CYP2D6HIF1ANFKB1
Tulobuterol SCHEMBL30986127 0.78 ADRB2 (1.00) ADRB2ADRB1CYP2D6HIF1ANFKB1
Flerobuterol SCHEMBL20819557 0.78 ADRB1 (0.66) ADRB2ADRB1CYP2D6HIF1ANFKB1
Tulobuterol SCHEMBL22970444 0.78 ADRB2 (1.00) ADRB2ADRB1CYP2D6HIF1ANFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110143886-B Process for the preparation of beta-arylaminoalkols such as tulobuterol, chlorpropaline, isoadrenaline dichloride and sotalol 北京化工大学 2022-11-01 CN disclosed
CN-110143886-A The method of the preparation such as beta-aromatic alkamine drug of tulobuterol, Clorprenaline, isoproterenol and Sotalol 北京化工大学 2019-08-20 CN disclosed