SCHEMBL28323720

SCHEMBL28323720

Clc1ccc(-c2c[nH]c3ncncc23)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA5 O75582 1/20 0.55
KIT P10721 2/20 0.54
JAK2 O60674 2/20 0.51
NTRK1 P04629 6/20 0.47
CDK2 P24941 2/20 0.46
CCNT1 O60563 1/20 0.46
CCNA2 P20248 1/20 0.46
CDK9 P50750 1/20 0.46
TNIK Q9UKE5 2/20 0.44
DYRK1A Q13627 3/20 0.44
AXL P30530 2/20 0.44
CLK1 P49759 2/20 0.44
DYRK2 Q92630 2/20 0.44
DYRK1B Q9Y463 2/20 0.44
PRKD3 O94806 2/20 0.44
MAP4K4 O95819 2/20 0.44
FLT4 P35916 2/20 0.44
KDR P35968 2/20 0.44
FLT3 P36888 2/20 0.44
FRK P42685 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23451864 0.78 CDK2 (0.53) KITJAK2NTRK1CDK2CCNT1
SCHEMBL27555122 0.78 CAMKK2 (0.49) RPS6KA5KITJAK2NTRK1CDK2
SCHEMBL25156923 0.76 TDO2 (0.67) RPS6KA5KITNTRK1DYRK1ADYRK2
SCHEMBL25193942 0.76 PIM1 (0.47) RPS6KA5KITNTRK1DYRK1ACLK1
SCHEMBL30407009 0.76 PIM1 (0.47) RPS6KA5KITNTRK1DYRK1ACLK1
SCHEMBL30349188 0.76 TDO2 (0.67) RPS6KA5KITNTRK1DYRK1ADYRK2
SCHEMBL858766 0.75 CAMKK2 (0.64) RPS6KA5KITJAK2CDK2CDK9
SCHEMBL21903027 0.73 RPS6KA5 (0.57) RPS6KA5JAK2NTRK1CDK9DYRK1A
SCHEMBL25208745 0.73 KIT (0.55) RPS6KA5KITJAK2NTRK1CDK2
SCHEMBL25518635 0.73 DYRK1A (0.45) RPS6KA5NTRK1TNIKDYRK1AAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110337294-A Pyrrolopyrimidines as CFTR potentiators 囊性纤维化基金会治疗公司 2019-10-15 CN disclosed