SCHEMBL28327682

SCHEMBL28327682

CC(C)(C)C(=O)ON1CC(NCc2ccc(Br)cc2N)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 8/20 0.36
USP30 Q70CQ3 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
HTT P42858 1/20 0.33
GRM2 Q14416 2/20 0.32
GRM3 Q14832 2/20 0.32
CARM1 Q86X55 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
LMNA P02545 1/20 0.32
GBA1 P04062 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CNR1 P21554 1/20 0.32
TBXA2R P21731 1/20 0.32
HRH2 P25021 1/20 0.32
SLC6A4 P31645 1/20 0.32
KCNH2 Q12809 1/20 0.32
HIF1A Q16665 1/20 0.32
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20045986 0.82 USP30 (0.48) AAK1USP30KRAS
SCHEMBL28328842 0.81 BCHE (0.41) MEN1KMT2AHTTCARM1PRMT6
SCHEMBL28566889 0.77 USP30 (0.55) USP30HTTKRAS
SCHEMBL28566888 0.77 USP30 (0.55) USP30HTTKRAS
SCHEMBL28777851 0.74 MEN1 (0.40) MEN1KMT2ACARM1PRMT6
SCHEMBL21874640 0.71 GRM2 (0.40) AAK1USP30KMT2AHTTGRM2
SCHEMBL21874641 0.71 GRM2 (0.40) AAK1USP30KMT2AHTTGRM2
SCHEMBL27945898 0.70 CARM1 (0.57) KMT2ACARM1PRMT6
Tert-Butyl Formate SCHEMBL28327683 0.70 SSTR4 (0.34) AAK1MEN1KMT2AHTTLMNA
SCHEMBL27765294 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110312711-A Heterocyclic compound and its application method as RAS inhibitor 亚瑞克西斯制药公司 2019-10-08 CN disclosed