SCHEMBL28327768

SCHEMBL28327768

O=CNC1CC(c2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.41
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
ADH1B P00325 4/20 0.39
ADH1A P07327 4/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C1 Q04828 1/20 0.39
TRPV1 Q8NER1 2/20 0.38
KAT2B Q92831 4/20 0.37
BRD9 Q9H8M2 1/20 0.37
ADH1C P00326 3/20 0.37
ADH7 P40394 2/20 0.37
SLC18A3 Q16572 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
ADH4 P08319 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14368356 0.82 GRIN2B (0.56) GRIN2BADH1BADH1AAKR1C3AKR1C1
SCHEMBL23130436 0.82 GRIN2B (0.56) GRIN2BADH1BADH1AAKR1C3AKR1C1
SCHEMBL28329005 0.81 ADRB2 (0.44) MAPTADH1BADH1AADH1CADH7
SCHEMBL14368359 0.81 ADRB2 (0.44) GRIN2BADH1BADH1ATRPV1ADH1C
SCHEMBL25994722 0.79 ADH1B (0.50) GAAMAPTADH1BADH1AADH1C
SCHEMBL25994590 0.79 ADH1B (0.50) GAAMAPTADH1BADH1AADH1C
SCHEMBL25994810 0.78 ESR1 (0.40) MAPTALDH1A1
SCHEMBL20653843 0.77 TRPV1 (0.48) AKR1C3AKR1C1TRPV1
SCHEMBL16762030 0.72 GAA (0.43) GRIN2BGAAMAPTAKR1C3AKR1C1
SCHEMBL16761873 0.72 GAA (0.43) GRIN2BGAAMAPTAKR1C3AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110461838-A oxadiazole transient receptor potential channel inhibitors HOFFMANN LA ROCHE 2019-11-15 CN disclosed