SCHEMBL28328124

SCHEMBL28328124

Brc1cc(-n2cccn2)nc(-n2cccn2)n1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.50
ADORA1 P30542 2/20 0.50
ADORA3 P0DMS8 1/20 0.50
ADORA2B P29275 1/20 0.50
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HTT P42858 2/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
G6PD P11413 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489646 0.79 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL28870957 0.76 HTT (0.62) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL29080878 0.75 NOTUM (0.48) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL2547816 0.72 ADORA2A (0.80) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL28186628 0.71 ALDH1A1 (0.55) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL9520789 0.70 KDM4E (0.50) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL6079917 0.70 ADORA2A (0.57) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL4289 0.70 KDM4E (0.50) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30261053 0.70 KDM4E (0.50) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL961121 0.69 ADORA2A (0.47) ADORA2AADORA1ADORA3ADORA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110290808-A 1- (the bromo- 6- of 4- amino -5- (1H- pyrazol-1-yl) pyrimidine -2-base) -1H- pyrazoles -4- alcohol and its purposes in treating cancer 诺华股份有限公司 2019-09-27 CN disclosed