SCHEMBL28328682

SCHEMBL28328682

O=C(O)Cc1c(-c2ccccc2)nnn1Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
ACHE P22303 1/20 0.42
BACE1 P56817 1/20 0.42
CFTR P13569 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ATM Q13315 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
PTK2 Q05397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28343059 0.86 IDO1 (0.51) KDM4EALDH1A1PTGDR2
SCHEMBL28328763 0.80 CYP19A1 (0.48) PTGDR2ADORA3
SCHEMBL28328678 0.80 PTGER4 (0.54) MEN1KMT2AALDH1A1PTGDR2ADORA3
SCHEMBL28329962 0.77 PTGDR2 (0.41) KDM4EPTGDR2
SCHEMBL28329954 0.76 CNR2 (0.48) ALDH1A1PTGDR2ATM
SCHEMBL11166536 0.74 PTGDR2 (0.49) MEN1KMT2AKDM4EALDH1A1PTGDR2
SCHEMBL11094843 0.74 PTGDR2 (0.52) MEN1KMT2AKDM4EALDH1A1PTGDR2
SCHEMBL28329955 0.73 PTGER4 (0.55) MEN1KMT2AKDM4EALDH1A1PTGDR2
SCHEMBL28329963 0.73 AKR1B1 (0.42) KDM4EALDH1A1PTGDR2
SCHEMBL6581989 0.71 TGM2 (0.51) TGM2MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110498773-B Method for synthesizing 1, 4-substituted 1,2, 3-triazole from acetylenic acid 乐山师范学院 2021-07-02 CN disclosed
CN-110526875-A A kind of acetylenic acid multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-12-03 CN disclosed
CN-110498772-A A kind of Terminal Acetylenes multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-110498773-A A kind of acetylenic acid synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-106866557-B (Z)-β-alkenyl bromine multicomponent prepares the method and application of 1,4- substitution -1,2,3- triazole 乐山师范学院 2019-11-12 CN disclosed