SCHEMBL28328678

SCHEMBL28328678

COc1ccc(Cn2nnc(-c3ccccc3)c2CC(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.54
AKR1C3 P42330 6/20 0.53
ERCC5 P28715 1/20 0.52
FEN1 P39748 1/20 0.52
PTGDR2 Q9Y5Y4 3/20 0.50
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HTT P42858 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ALOX15 P16050 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
TOP2A P11388 1/20 0.46
ALDH1A1 P00352 1/20 0.45
NPBWR1 P48145 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28343059 0.87 IDO1 (0.51) PTGER4PTGDR2SMN1; SMN2ALDH1A1
SCHEMBL15946997 0.82 PTGER4 (0.66) PTGER4AKR1C3ERCC5FEN1MEN1
SCHEMBL28328763 0.81 CYP19A1 (0.48) PTGER4PTGDR2ADORA3
SCHEMBL28329962 0.81 PTGDR2 (0.41) PTGER4PTGDR2HTTSMN1; SMN2
SCHEMBL28328682 0.80 TGM2 (0.44) PTGDR2MEN1KMT2AADORA3ALDH1A1
SCHEMBL11254519 0.78 PTGDR2 (0.60) PTGDR2MEN1KMT2AHTTSMN1; SMN2
SCHEMBL28329954 0.77 CNR2 (0.48) PTGDR2HTTSMN1; SMN2NPSR1L3MBTL1
SCHEMBL19927471 0.74 PTGS2 (0.56) PTGDR2NPSR1L3MBTL1ALDH1A1
SCHEMBL28329955 0.74 PTGER4 (0.55) PTGER4AKR1C3PTGDR2MEN1KMT2A
SCHEMBL6501472 0.74 ALDH1A1 (0.59) AKR1C3ERCC5FEN1PTGDR2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110498773-B Method for synthesizing 1, 4-substituted 1,2, 3-triazole from acetylenic acid 乐山师范学院 2021-07-02 CN disclosed
CN-110526875-A A kind of acetylenic acid multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-12-03 CN disclosed
CN-110498772-A A kind of Terminal Acetylenes multicomponent synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-110498773-A A kind of acetylenic acid synthesis 1,4- replaces the method for 1,2,3- triazole UNIV LESHAN NORMAL 2019-11-26 CN disclosed
CN-106866557-B (Z)-β-alkenyl bromine multicomponent prepares the method and application of 1,4- substitution -1,2,3- triazole 乐山师范学院 2019-11-12 CN disclosed