SCHEMBL28333752

SCHEMBL28333752

CCOc1ccc(C(=S)NCC(=O)OC)cc1OCC1CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
APOBEC3G Q9HC16 2/20 0.53
PDE4B Q07343 12/20 0.50
PDE4A P27815 6/20 0.50
PDE4C Q08493 6/20 0.50
PDE4D Q08499 6/20 0.50
ALDH1A1 P00352 2/20 0.50
HPGD P15428 1/20 0.50
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28333806 0.91 PDE4B (0.57) PDE4BPDE4APDE4CPDE4D
SCHEMBL28333853 0.89 PDE4B (0.60) PDE4BPDE4APDE4CPDE4DALDH1A1
SCHEMBL28334312 0.87 PDE4B (0.49) APOBEC3GPDE4BPDE4APDE4CPDE4D
SCHEMBL28634406 0.86 PDE4B (0.64) PDE4BPDE4APDE4CPDE4D
SCHEMBL17204895 0.85 TP53 (0.57) APOBEC3GPDE4BPDE4APDE4CPDE4D
SCHEMBL28033773 0.81 PDE4B (0.55) APOBEC3GPDE4BPDE4APDE4CPDE4D
SCHEMBL28333735 0.79 PDE4B (0.69) PDE4BPDE4APDE4CPDE4DPOLB
SCHEMBL28034335 0.78 TSHR (0.64) APOBEC3GPDE4BPDE4APDE4CPDE4D
SCHEMBL28034364 0.77 MAPK1 (0.65) PDE4BPDE4APDE4CPDE4DTSHR
SCHEMBL28034531 0.77 TP53 (0.63) ALDH1A1HPGDKDM4ETSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085429-B Aromatic heterocyclic derivative and application thereof in medicines 广东东阳光药业有限公司 2019-12-10 CN disclosed