SCHEMBL28337754

SCHEMBL28337754

COc1cccc(-c2cnc(N)nc2N)c1OC

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.52
MGAM O43451 1/20 0.48
GAA P10253 1/20 0.48
SI P14410 1/20 0.48
MGAM2 Q2M2H8 1/20 0.48
MEN1 O00255 1/20 0.46
SLC22A1 O15245 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP3A4 P08684 1/20 0.46
TSHR P16473 1/20 0.46
NFKB1 P19838 1/20 0.46
CYP2C19 P33261 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
DCPS Q96C86 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3948736 0.86 DHFR (0.54) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL4335673 0.86 DHFR (0.56) DHFRGAAALDH1A1
SCHEMBL4484811 0.85 DHFR (0.56) DHFRDCPS
SCHEMBL27805710 0.79 PIK3CD (0.51) MGAMGAASIMGAM2MEN1
SCHEMBL21223532 0.78 GAA (0.50) MGAMGAASIMGAM2ALDH1A1
SCHEMBL29398987 0.77 MGAM (0.49) DHFRMGAMGAASIMGAM2
SCHEMBL15673089 0.77 MGAM (0.49) DHFRMGAMGAASIMGAM2
SCHEMBL15672918 0.76 MGAM (0.51) MGAMGAASIMGAM2MEN1
SCHEMBL196440 0.76 MGAM (0.55) MGAMGAASIMGAM2ALDH1A1
SCHEMBL30507427 0.76 DYRK1A (0.60) MGAMGAASIMGAM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110325516-A HETEROARYL COMPOUNDS AND THEIR USE 米尼奥尔克斯治疗有限公司 2019-10-11 CN disclosed