SCHEMBL28339239

SCHEMBL28339239

NC(=O)c1cccn1NC(=O)[C@@H]1CC[C@H]1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
RAB9A P51151 3/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
GAA P10253 1/20 0.37
TAAR1 Q96RJ0 2/20 0.36
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPC1 O15118 1/20 0.36
KDM4E B2RXH2 3/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35
GRK2 P25098 1/20 0.35
CASP6 P55212 1/20 0.35
CASP8 Q14790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28339241 1.00 PARP1 (0.37) PARP1PARP10RAB9AMAPTLMNA
SCHEMBL3313426 0.80 SLC6A2 (0.36) RAB9AKMT2ANPC1KDM4E
SCHEMBL3313422 0.80 SLC6A2 (0.36) RAB9AKMT2ANPC1KDM4E
SCHEMBL9913081 0.80 SLC6A2 (0.36) RAB9AKMT2ANPC1KDM4E
SCHEMBL17174644 0.79 CYP2C19 (0.46) RAB9AMAPTLMNAGAAALDH1A1
SCHEMBL3312267 0.75 MAPK1 (0.39) ALDH1A1CYP2C19KDM4EHTTSMN1; SMN2
SCHEMBL1298778 0.72 LMNA (0.38) RAB9ALMNAALDH1A1L3MBTL1NPC1
SCHEMBL2060019 0.72 LMNA (0.38) PARP1MAPTLMNAALDH1A1L3MBTL1
SCHEMBL15956594 0.68 LMNA (0.42) RAB9AMAPTLMNAALDH1A1MEN1
SCHEMBL3311103 0.68 LMNA (0.36) RAB9ALMNACYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110627795-A Phosphodiesterase inhibitors and uses thereof 南京药捷安康生物科技有限公司 2019-12-31 CN disclosed