SCHEMBL2834138

SCHEMBL2834138

CC(C)(C)c1cc(-c2ccccc2)c2c(c1)C(O)(C(F)(F)F)C(=O)O2.CC(C)(C)c1ccc(O)c(-c2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.56
GABBR1 Q9UBS5 1/20 0.56
GPR84 Q9NQS5 1/20 0.36
ALDH1A1 P00352 3/20 0.34
NPC1 O15118 1/20 0.34
PLA2G1B P04054 1/20 0.34
NFKB1 P19838 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ATG4B Q9Y4P1 1/20 0.34
PDK2 Q15119 3/20 0.33
HSD17B2 P37059 1/20 0.32
CYP2D6 P10635 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826349 0.92 GABBR2 (0.64) GABBR2GABBR1GPR84ALDH1A1NPC1
SCHEMBL2826346 0.92 GABBR2 (0.64) GABBR2GABBR1GPR84ALDH1A1NPC1
SCHEMBL2826352 0.92 GABBR2 (0.64) GABBR2GABBR1GPR84ALDH1A1NPC1
SCHEMBL2828609 0.79 GABBR2 (0.81) GABBR2GABBR1ALDH1A1NPC1RAB9A
SCHEMBL3418225 0.74 BACE1 (0.56) ALDH1A1NPC1PLA2G1BNFKB1CASP3
SCHEMBL2371847 0.72 GABBR2 (1.00) GABBR2GABBR1
SCHEMBL2371842 0.72 GABBR2 (1.00) GABBR2GABBR1
SCHEMBL2371840 0.72 GABBR2 (1.00) GABBR2GABBR1
SCHEMBL4598293 0.68 GABBR2 (0.46) GABBR2GABBR1PDK2PTPN5
SCHEMBL30504387 0.66 KMT2A (0.52) ALDH1A1NPC1PLA2G1BNFKB1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1915357-B1 2-HYDROXY-PROPIONIC ACID DERIVATIVES AND 3-HYDROXY-BENZOFURAN-2-ONE DERIVATIVES WITH AFFINITY FOR THE GABA-B-RECEPTOR HOFFMANN LA ROCHE (CH) 2010-09-08 EP disclosed