SCHEMBL28341822

SCHEMBL28341822

Cn1cc(C(N)=O)c(=O)cc1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.47
CDK8 P49336 1/20 0.47
PKM P14618 1/20 0.43
MAP2K1 Q02750 9/20 0.38
MAP2K2 P36507 8/20 0.38
KDM4E B2RXH2 3/20 0.36
BRD4 O60885 2/20 0.36
ALDH1A1 P00352 1/20 0.36
BRPF1 P55201 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BRD9 Q9H8M2 1/20 0.35
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15991636 0.82 CCNC (0.49) CCNCCDK8PKMKDM4EBRD4
SCHEMBL29812644 0.81 MAP2K1 (0.41) MAP2K1MAP2K2KDM4EBRD4ALDH1A1
SCHEMBL23772011 0.78 L3MBTL1 (0.39) MAP2K1MAP2K2KDM4EBRD4BRD9
SCHEMBL29868687 0.77 MAP2K1 (0.41) MAP2K1MAP2K2KDM4E
SCHEMBL28838264 0.77 ADRA1D (0.36) CCNCCDK8
SCHEMBL19151400 0.74 CCNC (0.51) CCNCCDK8PKMMAP2K1MAP2K2
SCHEMBL13527129 0.74 CCNC (0.51) CCNCCDK8PKMKDM4EBRD4
SCHEMBL10002537 0.74 CDK8 (0.51) CCNCCDK8PKMMAP2K1MAP2K2
Hydrochloric Acid SCHEMBL17781591 0.72 CCNC (0.50) CCNCCDK8PKMKDM4EBRD4
SCHEMBL28811450 0.72 CCNC (0.50) CCNCCDK8PKMKDM4EBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110627796-B Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2022-07-12 CN disclosed
CN-110627796-A Nitrogenous heterocyclic derivative and application thereof in medicine 北京越之康泰生物医药科技有限公司 2019-12-31 CN disclosed
CN-110520416-A Polysubstituted pyridine ketones derivant, preparation method and its medical usage BEIJING YUEZHIKANGTAI BIOMEDICINES CO LTD 2019-11-29 CN disclosed