SCHEMBL28345159

SCHEMBL28345159

CC(C)(C)OC(=O)N(Cc1ccc(S)cc1)[C@H]1C[C@@H](C(=O)[O-])N(Cc2ccccc2Cl)C1.[H+]

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.40
NR1H4 Q96RI1 1/20 0.37
KDM1A O60341 3/20 0.35
NPFFR1 Q9GZQ6 2/20 0.34
NPFFR2 Q9Y5X5 2/20 0.34
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
SLC16A3 O15427 4/20 0.33
SLC16A1 P53985 4/20 0.33
MCTS1 Q9ULC4 3/20 0.33
REN P00797 1/20 0.33
GAA P10253 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
S1PR1 P21453 1/20 0.33
S1PR5 Q9H228 1/20 0.33
GRM2 Q14416 1/20 0.32
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28348072 0.92 HSD11B1 (0.42) HSD11B1NR1H4KDM1ANPFFR1NPFFR2
SCHEMBL28348073 0.82 NPFFR1 (0.45) HSD11B1NR1H4NPFFR1NPFFR2SLC16A3
SCHEMBL29930557 0.81 NPFFR1 (0.50) HSD11B1NR1H4NPFFR1NPFFR2SLC16A3
SCHEMBL29930039 0.80 ATM (0.41) HSD11B1NR1H4KDM1ANPFFR1NPFFR2
SCHEMBL2824379 0.76 HSD11B1 (0.52) HSD11B1NR1H4JAK2JAK1KMT2A
SCHEMBL13841892 0.76 HSD11B1 (0.52) HSD11B1NR1H4JAK2JAK1KMT2A
SCHEMBL2822792 0.74 HSD11B1 (0.50) HSD11B1NR1H4KDM1AHDAC8HDAC6
SCHEMBL13841889 0.74 HSD11B1 (0.50) HSD11B1NR1H4KDM1AHDAC8HDAC6
SCHEMBL26966069 0.69 HSD11B1 (0.52) HSD11B1NR1H4JAK2JAK1
SCHEMBL2819571 0.67 HTR2A (0.46) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110546136-A proline-based neuropeptide FF receptor modulators RES TRIANGLE INST 2019-12-06 CN disclosed