SCHEMBL28355488

SCHEMBL28355488

O=C(O)c1ccc(C(=O)N2CCCCC2)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 2/20 0.54
HPGD P15428 8/20 0.53
ALDH1A1 P00352 1/20 0.53
CNR1 P21554 3/20 0.51
USP2 O75604 1/20 0.49
TSHR P16473 3/20 0.48
POLB P06746 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29606862 1.00 CPS1 (0.54) CPS1HPGDALDH1A1CNR1USP2
SCHEMBL28351918 0.82 CPS1 (0.59) CPS1HPGDALDH1A1TSHRMEN1
SCHEMBL29816274 0.82 CNR1 (0.63) CPS1HPGDALDH1A1CNR1USP2
Hydrochloric Acid SCHEMBL28469010 0.81 CNR1 (0.61) CPS1HPGDALDH1A1CNR1USP2
SCHEMBL5096987 0.81 HPGD (0.55) HPGDALDH1A1TSHRPOLBKMT2A
SCHEMBL1355120 0.80 HPGD (0.56) CPS1HPGDALDH1A1TSHRPOLB
SCHEMBL12205464 0.79 CPS1 (0.58) CPS1HPGDALDH1A1CNR1USP2
SCHEMBL5110700 0.79 POLB (0.66) HPGDALDH1A1USP2TSHRPOLB
SCHEMBL5103701 0.79 L3MBTL3 (0.62) HPGDALDH1A1TSHRPOLBMEN1
SCHEMBL969401 0.79 CCKBR (0.58) CPS1HPGDALDH1A1CNR1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110759889-B 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2022-05-20 CN disclosed
CN-110759889-A 2-aryl amido substituted thiophene imide ester compound and preparation method and application thereof 中国医学科学院药物研究所 2020-02-07 CN disclosed