SCHEMBL28356002

SCHEMBL28356002

CCOC(c1ccccc1)c1cnc(-c2ccccc2)n1-c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
MDM2 Q00987 1/20 0.41
PLK1 P53350 1/20 0.41
CACNA2D1 P54289 1/20 0.41
FNTA P49354 2/20 0.40
FNTB P49356 2/20 0.40
LMNA P02545 3/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
VCP P55072 1/20 0.39
TP53 P04637 2/20 0.38
THRB P10828 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28352526 0.89 PLK1 (0.39) PLK1HPGDKDM4EALDH1A1TP53
SCHEMBL28356556 0.88 HPGD (0.47) GABRA2GABRB2CACNA2D1LMNAHPGD
SCHEMBL28352367 0.87 GLA (0.43) GABRA2GABRB2CACNA2D1LMNAHPGD
SCHEMBL28355861 0.87 TSHR (0.40) GABRA2GABRB2CACNA2D1HPGDTP53
SCHEMBL28356404 0.87 DCTPP1 (0.41) CACNA2D1LMNAHPGDALDH1A1VCP
SCHEMBL28356151 0.85 HPGD (0.40) PLK1CACNA2D1HPGDALDH1A1TP53
SCHEMBL28352441 0.84 MDM2 (0.43) GABRA2GABRB2MDM2PLK1CACNA2D1
SCHEMBL28356409 0.82 HPGD (0.42) PLK1CACNA2D1HPGDKDM4EALDH1A1
SCHEMBL28352337 0.81 HPGD (0.43) GABRA2GABRB2PLK1CACNA2D1HPGD
SCHEMBL28356143 0.81 CACNA2D1 (0.41) PLK1CACNA2D1HPGDALDH1A1VCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107162982-B Imidazole compounds with anticancer activity and derivatives thereof 广东药科大学 2020-02-11 CN disclosed