SCHEMBL28358149

SCHEMBL28358149

O=C(O)CNC(=O)/C=C/c1cn(-c2ccccc2)nc1-c1ccc2ccccc2c1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 1/20 0.58
HDAC1 Q13547 12/20 0.54
HDAC2 Q92769 12/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
PTPN2 P17706 1/20 0.52
PTPN1 P18031 1/20 0.52
PTPN6 P29350 1/20 0.52
CDC25B P30305 1/20 0.52
PTPN11 Q06124 1/20 0.52
RAB9A P51151 1/20 0.52
NPSR1 Q6W5P4 1/20 0.51
RAD52 P43351 1/20 0.51
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29051092 1.00 MAPT (0.58) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL28361894 0.89 MAPT (0.57) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL28358299 0.85 MEN1 (0.74) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL28361850 0.85 MEN1 (0.74) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL28358398 0.85 MEN1 (0.74) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL29051128 0.84 MEN1 (0.52) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL28361829 0.84 MEN1 (0.52) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL29051131 0.84 MEN1 (0.52) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL30511846 0.83 KDM4E (0.69) MAPTKDM4EALDH1A1HDAC1HDAC2
SCHEMBL29051122 0.82 MEN1 (0.53) MAPTKDM4EALDH1A1HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110746355-A Phenylpyrazole compound, pharmaceutical composition, preparation method and application thereof 中国科学院上海有机化学研究所 2020-02-04 CN claimed
CN-110746355-B Phenylpyrazole compound, pharmaceutical composition, and preparation method and application thereof 中国科学院上海有机化学研究所 2023-08-11 CN disclosed
CN-110746355-A Phenylpyrazole compound, pharmaceutical composition, preparation method and application thereof 中国科学院上海有机化学研究所 2020-02-04 CN disclosed