SCHEMBL28358908

SCHEMBL28358908

O=C(Nc1c(I)cc(Br)cc1[N+](=O)[O-])C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ERN1 O75460 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AR P10275 3/20 0.35
PGR P06401 1/20 0.35
CYP3A4 P08684 1/20 0.35
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AKR1C2 P52895 1/20 0.34
AKR1C1 Q04828 1/20 0.34
PARP1 P09874 1/20 0.33
GPR35 Q9HC97 1/20 0.33
FBP1 P09467 1/20 0.33
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15985062 0.83 ALDH1A1 (0.44) GAAMAPK1ERN1MEN1KMT2A
SCHEMBL28549978 0.81 AR (0.38) GAAMAPK1RXFP1ERN1MEN1
SCHEMBL31248747 0.80 AR (0.38) GAAMAPK1RXFP1ERN1MEN1
SCHEMBL28362640 0.79 VCAM1 (0.42) MAPK1RXFP1MEN1KMT2ASMN1; SMN2
SCHEMBL220261 0.79 PDGFRB (0.38) MEN1KMT2AARPGRCYP3A4
SCHEMBL28362551 0.77 VCAM1 (0.46) MAPK1MEN1KMT2APGRCYP3A4
SCHEMBL31312674 0.77 ALDH1A1 (0.39) SMN1; SMN2
SCHEMBL28362598 0.76 MAPK1 (0.37) GAAMAPK1RXFP1ERN1AR
SCHEMBL7784821 0.76 HRAS (0.41) GAAMAPK1RXFP1MEN1KMT2A
SCHEMBL10322564 0.75 ALDH1A1 (0.38) MAPK1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248472-B Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2022-06-28 CN disclosed
CN-113248472-A Anti-osteoporosis compound and derivative thereof, pharmaceutical composition, preparation method and application 中国药科大学 2021-08-13 CN disclosed
CN-110818609-A Preparation method and application of 3-acetyl indole BRPF1 inhibitor 中国药科大学 2020-02-21 CN disclosed