SCHEMBL28359571

SCHEMBL28359571

CC(C)(C)[C@](C)(C(=O)O)N1Cc2ccc(Br)cc2C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SDCBP O00560 1/20 0.36
SDC2 P34741 1/20 0.36
CUL4A Q13619 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA6 Q16445 1/20 0.35
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
HSD17B3 P37058 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23309876 1.00 MEN1 (0.36) MEN1KMT2ASDCBPSDC2CUL4A
SCHEMBL18793920 0.82 MEN1 (0.41) MEN1KMT2ACUL4AGABRA1GABRG2
SCHEMBL19475669 0.82 HSD17B3 (0.39) MEN1KMT2ASDCBPSDC2GABRA1
SCHEMBL2178347 0.80 GABRA1 (0.36) MEN1KMT2ASDCBPSDC2CUL4A
SCHEMBL18765683 0.78 GABRA1 (0.43) MEN1KMT2ACUL4AGABRA1GABRG2
SCHEMBL16099526 0.77 SDCBP (0.47) MEN1KMT2ASDCBPSDC2HSD17B3
SCHEMBL23309869 0.75 ROCK1 (0.39)
SCHEMBL17141692 0.71 PIK3CA (0.46) MEN1KMT2AGABRA1GABRG2GABRB3
SCHEMBL29507022 0.71 MEN1 (0.59) MEN1KMT2ACUL4AGABRA1GABRG2
SCHEMBL290015 0.71 MEN1 (0.59) MEN1KMT2ACUL4AGABRA1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110831939-A 6-pyrimidine-isoindole derivatives as ERK1/2 inhibitors 大冢制药株式会社 2020-02-21 CN disclosed