SCHEMBL28360398

SCHEMBL28360398

Nc1cnc(N(c2ccccc2)c2ccccc2)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.52
ALDH1A1 P00352 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
TSHR P16473 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
NPC1 O15118 1/20 0.43
JAK2 O60674 1/20 0.43
RAB9A P51151 1/20 0.43
SYK P43405 1/20 0.42
HDAC6 Q9UBN7 4/20 0.41
HDAC1 Q13547 3/20 0.41
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28504853 0.79 HDAC6 (0.49) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL4582422 0.79 TDP1 (0.54) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL18294910 0.78 ALDH1A1 (0.45) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL21943233 0.75 HDAC6 (0.51) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL6879552 0.74 ALDH1A1 (0.55) ALDH1A1TDP1KDM4ETSHRHDAC6
SCHEMBL16675141 0.74 HDAC6 (0.44) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL4399532 0.73 ALDH1A1 (0.48) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL16483989 0.71 ALDH1A1 (0.47) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL183387 0.71 MAPT (0.70) MAPTALDH1A1TDP1L3MBTL1KDM4E
SCHEMBL18294907 0.71 HDAC6 (0.51) MAPTALDH1A1TDP1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141123-B Compound, preparation method thereof and application thereof in preparation of dual inhibitors of histone deacetylase and epoxide hydrolase 沈阳药科大学 2024-05-17 CN disclosed
CN-115141123-A Compound, preparation method thereof and application thereof in preparation of histone deacetylase and epoxide hydrolase dual inhibitor 沈阳药科大学 2022-10-04 CN disclosed
CN-110835406-B Free radical monomer containing diphenylamine structure and preparation method and application of polymer thereof 武汉理工大学 2020-09-01 CN disclosed
CN-110835406-A Novel free radical monomer containing diphenylamine structure and preparation method and application of polymer thereof 武汉理工大学 2020-02-25 CN disclosed