SCHEMBL28360809

SCHEMBL28360809

COc1ccc(C=CC(=O)C=Cc2ccc(O)cc2)c(OC)c1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 1/20 0.85
CTSB P07858 1/20 0.85
BACE1 P56817 3/20 0.81
MAPT P10636 4/20 0.78
MEN1 O00255 2/20 0.78
KMT2A Q03164 2/20 0.78
ALDH1A1 P00352 1/20 0.78
STAT3 P40763 1/20 0.67
XDH P47989 1/20 0.66
CHRNA7 P36544 1/20 0.63
NFKB1 P19838 2/20 0.62
DPP4 P27487 1/20 0.62
NFKB2 Q00653 1/20 0.62
RELA Q04206 1/20 0.62
NPC1 O15118 1/20 0.62
MAPK1 P28482 1/20 0.62
RAB9A P51151 1/20 0.62
JUN P05412 1/20 0.61
F3 P13726 1/20 0.60
TXNRD1 Q16881 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3204166 0.90 BACE1 (1.00) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL3204181 0.90 BACE1 (1.00) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL5598357 0.89 MAPT (1.00) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL5598355 0.89 MAPT (1.00) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL1976945 0.86 CYP1A2 (0.81) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL18508908 0.85 MAPT (0.81) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL28609815 0.84 F3 (0.86) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL28838366 0.83 MAPT (0.67) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL7180313 0.82 TNFRSF1A (0.86) CAPN1CTSBBACE1MAPTMEN1
SCHEMBL29600833 0.82 TNFRSF1A (0.86) CAPN1CTSBBACE1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114634465-B Pentadienone derivative containing sulfonyl piperazine as well as preparation method and application thereof 贵州大学 2023-05-30 CN disclosed
CN-114634465-A Sulfonyl piperazine-containing pentadiene ketone derivative and preparation method and application thereof 贵州大学 2022-06-17 CN disclosed
CN-108530435-B Quinoxaline-containing 1, 4-pentadiene-3-ketone derivative, preparation method and application 贵州大学 2021-08-17 CN disclosed
CN-106928176-B Coumarin-containing 1, 4-pentadiene-3-ketone derivative and preparation method and application thereof 贵州大学 2020-02-18 CN disclosed