SCHEMBL28838366

SCHEMBL28838366

COc1ccc(C=CC(=O)C=Cc2ccc(OCCBr)cc2)c(OC)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.67
ALDH1A1 P00352 2/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
CAPN1 P07384 1/20 0.63
CTSB P07858 1/20 0.63
BACE1 P56817 1/20 0.61
HDAC8 Q9BY41 4/20 0.57
TXNRD1 Q16881 1/20 0.54
TXNRD3 Q86VQ6 1/20 0.54
TXNRD2 Q9NNW7 1/20 0.54
JUN P05412 1/20 0.53
NFKB1 P19838 1/20 0.53
LY96 Q9Y6Y9 1/20 0.53
APP P05067 1/20 0.53
F3 P13726 1/20 0.52
CYP1A1 P04798 1/20 0.52
CYP1A2 P05177 1/20 0.52
NFE2L2 Q16236 1/20 0.52
CYP1B1 Q16678 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28838351 0.86 F3 (0.71) MAPTKMT2ACAPN1CTSBBACE1
SCHEMBL29575068 0.85 TNFRSF1A (0.74) MAPTALDH1A1MEN1KMT2ACTSB
SCHEMBL28838374 0.84 GSK3B (0.59) MAPTALDH1A1MEN1KMT2AHDAC8
SCHEMBL28360809 0.83 CAPN1 (0.85) MAPTALDH1A1MEN1KMT2ACAPN1
SCHEMBL5598355 0.82 MAPT (1.00) MAPTALDH1A1MEN1KMT2ACAPN1
SCHEMBL5598357 0.82 MAPT (1.00) MAPTALDH1A1MEN1KMT2ACAPN1
SCHEMBL18508908 0.79 MAPT (0.81) MAPTALDH1A1MEN1KMT2ACAPN1
SCHEMBL28838354 0.79 PPARA (0.56) MAPTKMT2ABACE1JUNF3
SCHEMBL28838365 0.78 MAPT (0.50) MAPTALDH1A1MEN1KMT2ACAPN1
SCHEMBL28838357 0.77 MAOB (0.55) MAPTALDH1A1MEN1KMT2ABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109721559-B 1, 4-pentadiene-3-ketone derivative containing thioether triazole, preparation method and application 贵州大学 2022-02-15 CN disclosed