SCHEMBL28364643

SCHEMBL28364643

CCC(C)(Cc1ccccc1)C(=O)NOc1cc(C)nn1-c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.42
LMNA P02545 1/20 0.41
STAT1 P42224 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 4/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
GAA P10253 2/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
ATM Q13315 1/20 0.40
PTGS2 P35354 1/20 0.40
P2RY1 P47900 1/20 0.40
TSHR P16473 1/20 0.39
KCNJ6 P48051 1/20 0.39
KCNJ5 P48544 1/20 0.39
KCNJ3 P48549 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21753619 0.83 NTRK1 (0.50) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL25285702 0.83 NTRK1 (0.43) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL21753616 0.78 ALDH1A1 (0.50) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL21753627 0.76 ALDH1A1 (0.48) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL21753629 0.73 P2RY1 (0.51) NTRK1LMNASTAT1ALDH1A1MAPT
SCHEMBL25285703 0.72 P2RY1 (0.44) NTRK1LMNASTAT1ALDH1A1MAPT
SCHEMBL28364642 0.72 ALDH1A1 (0.42) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL21753652 0.71 KMT2A (0.51) NTRK1LMNASTAT1ALDH1A1MAPT
SCHEMBL21753656 0.71 ALDH1A1 (0.46) NTRK1LMNASTAT1ALDH1A1HTT
SCHEMBL21753653 0.71 P2RY1 (0.48) NTRK1ALDH1A1MAPTL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110857285-B Substituted pyrazole compound, preparation method, pharmaceutical composition and application thereof 江苏万高药业股份有限公司 2022-12-20 CN disclosed
CN-110857285-A Substituted pyrazole compound, preparation method, pharmaceutical composition and application thereof 天津谷堆生物医药科技有限公司 2020-03-03 CN disclosed