SCHEMBL28366232

SCHEMBL28366232

O=c1c2cc([N+](=O)[O-])ccc2ccn1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.45
PHOSPHO1 Q8TCT1 1/20 0.42
MIF P14174 1/20 0.41
G6PD P11413 1/20 0.40
TLR9 Q9NR96 1/20 0.40
MEN1 O00255 2/20 0.39
POLB P06746 2/20 0.39
KMT2A Q03164 2/20 0.39
SLC6A9 P48067 1/20 0.39
SLC6A5 Q9Y345 1/20 0.39
MAPT P10636 1/20 0.39
RECQL P46063 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM1A O60341 1/20 0.38
ALOX5 P09917 1/20 0.38
PTGS2 P35354 1/20 0.38
NOX1 Q9Y5S8 1/20 0.38
ENPP2 Q13822 1/20 0.37
CDC7 O00311 1/20 0.37
PTPN1 P18031 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28366388 0.88 TNF (0.45) KIF11PHOSPHO1G6PDTLR9SLC6A9
SCHEMBL16862008 0.80 KCNH2 (0.48) KIF11MEN1POLBKMT2ASLC6A9
SCHEMBL14966623 0.79 NPC1 (0.44) KIF11PHOSPHO1MIFMEN1POLB
SCHEMBL28366314 0.79 LCK (0.43) KIF11PHOSPHO1MIFG6PDTLR9
Trifluoromethanesulfonic Acid SCHEMBL27781891 0.78 POLB (0.38) PHOSPHO1MEN1POLBKMT2AMAPT
SCHEMBL28057350 0.77 ALDH1A1 (0.49) PHOSPHO1MIFG6PDTLR9MEN1
SCHEMBL9920084 0.75 MEN1 (0.55) MEN1POLBKMT2AMAPTPLEC
SCHEMBL31285936 0.75 TRPV1 (0.51) PHOSPHO1G6PDTLR9MAPT
SCHEMBL4648405 0.73 POLB (0.39) MIFMEN1POLBKMT2AMAPT
SCHEMBL2611447 0.73 HDAC8 (0.40) MEN1POLBKMT2AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105523996-B Amide derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2020-03-06 CN disclosed