SCHEMBL28374362

SCHEMBL28374362

COn1cc(CC(=O)Nc2ccccc2F)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.54
ALDH1A1 P00352 3/20 0.51
HTT P42858 2/20 0.51
HPGD P15428 2/20 0.51
POLB P06746 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
RCE1 Q9Y256 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
S1PR2 O95136 2/20 0.49
MAPT P10636 1/20 0.49
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 2/20 0.47
PARP1 P09874 1/20 0.47
PKM P14618 1/20 0.46
TP53 P04637 2/20 0.46
BRD4 O60885 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28369737 0.86 PTPN5 (0.51) TSHRALDH1A1HTTPOLBS1PR2
SCHEMBL28373077 0.85 S1PR2 (0.57) TSHRALDH1A1HTTPOLBL3MBTL1
SCHEMBL28369732 0.85 S1PR2 (0.49) TSHRALDH1A1HTTPOLBS1PR2
SCHEMBL28369520 0.85 S1PR2 (0.49) TSHRALDH1A1HTTS1PR2MAPT
SCHEMBL28375685 0.85 S1PR2 (0.57) TSHRALDH1A1HTTS1PR2MAPT
SCHEMBL28167902 0.84 KDM4E (0.57) TSHRALDH1A1HTTHPGDPOLB
SCHEMBL28375698 0.84 PTPN5 (0.56) TSHRALDH1A1HTTPOLBS1PR2
SCHEMBL28373924 0.84 ALDH1A1 (0.57) TSHRALDH1A1HTTHPGDPOLB
SCHEMBL28885207 0.81 MAPT (0.52) TSHRALDH1A1POLBS1PR2MAPT
SCHEMBL28369364 0.80 MAPT (0.57) ALDH1A1S1PR2MAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107149602-B Application of indole compounds and derivatives thereof in preparation of anti-HIV drugs 中国医学科学院药物研究所 2020-10-09 CN disclosed
CN-107149603-B Application of indole compounds and derivatives thereof in preparation of anti-influenza virus drugs 中国医学科学院药物研究所 2020-07-14 CN disclosed
CN-107176921-B Indole compounds with antiviral activity in isatis root and derivatives thereof 中国医学科学院药物研究所 2020-03-31 CN disclosed