SCHEMBL28375855

SCHEMBL28375855

COc1cc2c3c(Cl)nccc3n(C(=O)O)c2cc1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
BRD4 O60885 3/20 0.34
BRD2 P25440 2/20 0.34
BRD3 Q15059 2/20 0.34
HTT P42858 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
PDE10A Q9Y233 1/20 0.34
PTGS2 P35354 2/20 0.33
PTGS1 P23219 1/20 0.33
KMO O15229 1/20 0.33
AURKB Q96GD4 2/20 0.33
CGAS Q8N884 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20581226 0.85 TLR9 (0.38) BRD4BRD2BRD3AURKBPOLB
SCHEMBL28373125 0.83 CYP1A2 (0.38) LMNAKDM4ECYP3A4MAPTHPGD
SCHEMBL28371735 0.82 QDPR (0.34) PDE10A
SCHEMBL20581859 0.82 SRD5A1 (0.47) HPGDMEN1KMT2AHDAC6
SCHEMBL28885625 0.81 KDM4E (0.38) LMNAKDM4EMAPTPOLBAURKA
SCHEMBL20581869 0.80 ERN1 (0.39) LMNAKDM4ECYP3A4MAPTHPGD
SCHEMBL28376323 0.80 CGAS (0.40) LMNAKDM4ECYP3A4MAPTHPGD
SCHEMBL28376695 0.80 EGFR (0.39) LMNAKDM4E
SCHEMBL28371632 0.79 DPP4 (0.35) PDE3BPDE3APDE10ACYP1A2HSP90AA1
SCHEMBL28375857 0.77 MAOA (0.39) LMNAKDM4ECYP3A4MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997671-A Azaindole compounds as histone methyltransferase inhibitors 全球血液疗法股份有限公司 2020-04-10 CN disclosed