SCHEMBL28378463

SCHEMBL28378463

O=C(NC1CC1)c1ccc(O)cc1Cl

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.69
NPC1 O15118 3/20 0.60
RAB9A P51151 3/20 0.60
P2RX7 Q99572 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.51
SLC6A12 P48065 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.49
TAS1R1 Q7RTX1 1/20 0.49
TAS1R2 Q8TE23 1/20 0.49
ALDH1A1 P00352 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
ESRRB O95718 1/20 0.46
ESRRG P62508 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA3 P07451 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29077678 0.85 HPGD (0.71) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL10282412 0.82 RAB9A (0.86) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL1820539 0.82 HPGD (0.68) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL4516890 0.82 HPGD (0.68) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL20056512 0.81 HPGD (0.62) HPGDNPC1RAB9AP2RX7SMN1; SMN2
Water SCHEMBL27924604 0.81 HPGD (0.66) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL12672349 0.81 HPGD (0.66) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL4043511 0.80 HPGD (0.64) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL22845271 0.78 HPGD (0.62) HPGDNPC1RAB9AP2RX7SMN1; SMN2
SCHEMBL104356 0.78 HPGD (0.62) HPGDNPC1RAB9AP2RX7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110818634-B Refining method of lervatinib mesylate 上海新礼泰药业有限公司 2021-11-30 CN disclosed
CN-110818634-A Refining method of lervatinib mesylate 上海博志研新药物技术有限公司 2020-02-21 CN disclosed