SCHEMBL28384635

SCHEMBL28384635

O=C(Nc1ccc(Cl)nn1)C1CC12CCN(C(=O)O)CC2

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.38
HTT P42858 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
LMNA P02545 2/20 0.34
ALDH1A1 P00352 2/20 0.34
EPHX2 P34913 1/20 0.34
NPY5R Q15761 1/20 0.34
LRRK2 Q5S007 3/20 0.33
POLB P06746 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KCNH2 Q12809 2/20 0.33
MARK3 P27448 1/20 0.33
SCN5A Q14524 1/20 0.33
MAP4K1 Q92918 1/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27008525 0.86 MAP4K1 (0.37) LMNAALDH1A1NPY5RLRRK2KCNH2
SCHEMBL20641873 0.85 NAMPT (0.43)
SCHEMBL31195181 0.81 FAAH (0.39) FAAHLMNAALDH1A1MAP4K1HPGD
SCHEMBL26619952 0.81 FAAH (0.39) FAAHLMNAALDH1A1MAP4K1HPGD
SCHEMBL27008482 0.78 EPHX2 (0.44) FAAHHTTNPC1RAB9ALMNA
SCHEMBL27008627 0.78 EPHX2 (0.44) FAAHHTTNPC1RAB9ALMNA
SCHEMBL27008496 0.77 SMN1; SMN2 (0.43) HTTNPC1RAB9ALMNAALDH1A1
SCHEMBL27008607 0.77 SMN1; SMN2 (0.43) HTTNPC1RAB9ALMNAALDH1A1
SCHEMBL27008487 0.77 HCRTR2 (0.50) HTTNPC1RAB9AALDH1A1EPHX2
SCHEMBL27008613 0.77 HCRTR2 (0.50) HTTNPC1RAB9AALDH1A1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110891569-A Antagonists of muscarinic acetylcholine receptor M4 范德堡大学 2020-03-17 CN disclosed