SCHEMBL28385754

SCHEMBL28385754

Cc1cc(Cl)nc2ccc(-c3ccc4nn(C)cc4c3)cc12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
HIF1A Q16665 1/20 0.49
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
BACE1 P56817 1/20 0.36
ALDH1A1 P00352 2/20 0.36
NSD2 O96028 1/20 0.36
MAPT P10636 1/20 0.36
CHRM1 P11229 5/20 0.35
HTT P42858 1/20 0.35
MAT2A P31153 1/20 0.35
NOTUM Q6P988 1/20 0.35
MAPK1 P28482 1/20 0.34
ADCY10 Q96PN6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31218441 0.83 KDM4E (0.41) KDM4EMAOAMAOBBACE1ALDH1A1
SCHEMBL20582309 0.83 KDM4E (0.41) KDM4EMAOAMAOBBACE1ALDH1A1
SCHEMBL22028370 0.81 LMNA (0.37) KDM4EBACE1ALDH1A1NSD2MAPT
SCHEMBL31218461 0.81 LMNA (0.37) KDM4EBACE1ALDH1A1NSD2MAPT
SCHEMBL7059007 0.77 KDM4E (0.58) KDM4ECYP3A4CYP2C19HIF1ABACE1
SCHEMBL22028368 0.75 MAOA (0.38) KDM4EMAOAMAOBBACE1CHRM1
SCHEMBL31218446 0.75 MAOA (0.38) KDM4EMAOAMAOBBACE1CHRM1
SCHEMBL22028265 0.74 TLR8 (0.44) BACE1HTTMAT2A
Hydrochloric Acid SCHEMBL28383603 0.74 TLR8 (0.43) HTTMAT2A
SCHEMBL29303290 0.72 KDM4E (0.42) KDM4EMAOAMAOBBACE1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111065626-B Compounds for the treatment of huntington's disease PTC医疗公司 2024-09-27 CN disclosed
CN-111065626-A Compounds for the treatment of huntington's chorea PTC医疗公司 2020-04-24 CN disclosed