SCHEMBL28386643

SCHEMBL28386643

NC(=S)NN=C1CCNc2cc(F)c(F)c(F)c21

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 14/20 0.52
ALDH1A1 P00352 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28387201 0.81 CTSL (0.64) CTSLALDH1A1L3MBTL1KDM4E
SCHEMBL28381906 0.74 CTSL (0.73) CTSLALDH1A1L3MBTL1KDM4ETDP1
SCHEMBL28284166 0.70 CTSL (0.67) CTSLALDH1A1L3MBTL1KDM4EMEN1
SCHEMBL28383150 0.68 CTSL (0.52) CTSLALDH1A1L3MBTL1KDM4EMEN1
SCHEMBL28887932 0.68 CTSL (0.73) CTSLALDH1A1L3MBTL1KDM4E
SCHEMBL6337478 0.68 CTSL (1.00) CTSLALDH1A1L3MBTL1KDM4E
SCHEMBL28382176 0.67 CTSL (0.53) CTSLALDH1A1L3MBTL1KDM4E
SCHEMBL18477265 0.67 CTSL (0.53) CTSLALDH1A1L3MBTL1KDM4EMEN1
SCHEMBL28388654 0.66 CTSL (0.58) CTSLALDH1A1L3MBTL1KDM4ELMNA
SCHEMBL28382175 0.66 MEN1 (0.39) ALDH1A1L3MBTL1KDM4EMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109503478-B 2, 3-dihydro-1H-quinoline-4-ketone thiosemicarbazone derivative and preparation method and application thereof 岭南师范学院 2020-04-24 CN disclosed