SCHEMBL28389605

SCHEMBL28389605

O=C=C1CCC(c2ccc(Br)cc2)C(O)(C(=O)O)C1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.33
RORC P51449 2/20 0.32
KDM1A O60341 3/20 0.32
RCOR1 Q9UKL0 3/20 0.32
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28389604 0.82 LIG1 (0.38) LIG1RORCKDM1ARCOR1HDAC4
SCHEMBL7969974 0.68 MAPK1 (0.38) KDM1A
SCHEMBL8031930 0.62 KDM1A (0.44) LIG1RORCKDM1ARCOR1HDAC4
Hydrochloric Acid SCHEMBL2075502 0.61 KDM1A (0.53) LIG1KDM1ARCOR1HDAC4
SCHEMBL7987943 0.60 PKM (0.34)
SCHEMBL11019711 0.60 HTR7 (0.40) LIG1RORCKDM1ARCOR1HDAC4
SCHEMBL4133969 0.60 KDM1A (0.44) LIG1RORCKDM1ARCOR1HDAC4
SCHEMBL15766917 0.59 KDM1A (0.51) LIG1RORCKDM1ARCOR1HDAC4
SCHEMBL12825788 0.59 MAPK1 (0.48) LIG1RORCKDM1ARCOR1HDAC4
SCHEMBL15766918 0.59 KDM1A (0.51) LIG1RORCKDM1ARCOR1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110938083-B Compounds as BACE1 inhibitors and uses thereof 南京圣和药业股份有限公司 2022-06-07 CN disclosed
CN-110938083-A Compounds as BACE1 inhibitors and uses thereof 南京圣和药业股份有限公司 2020-03-31 CN disclosed