SCHEMBL28393152

SCHEMBL28393152

C#CCOc1cccc(OCc2cccnc2)c1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.53
GPR132 Q9UNW8 12/20 0.47
CMKLR2 P46091 1/20 0.46
CMKLR1 Q99788 1/20 0.46
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
CYP11B1 P15538 1/20 0.45
MAOB P27338 1/20 0.45
GRM2 Q14416 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28011530 0.88 MAPK1 (0.64) MAPK1GPR132CMKLR2CMKLR1HTR1A
SCHEMBL28397433 0.84 NOS3 (0.51) MAPK1GPR132MAOB
SCHEMBL28397085 0.82 MAPK1 (0.42) MAPK1HTR1ADRD2CYP11B1
SCHEMBL28396007 0.82 MAOB (0.62) MAOB
SCHEMBL791886 0.81 MAOB (0.66) MAPK1GPR132HTR1ADRD2MAOB
SCHEMBL4808799 0.80 CHRNB2 (0.51) MAOB
SCHEMBL22964344 0.79 MAPK1 (0.58) MAPK1GPR132CMKLR2CMKLR1
SCHEMBL21477258 0.78 MAPK1 (0.57) MAPK1GPR132CMKLR2CMKLR1HTR1A
SCHEMBL3998456 0.78 MAOB (0.66) MAPK1GPR132CMKLR2CMKLR1CYP11B1
SCHEMBL13452125 0.78 MAPK1 (0.57) MAPK1GPR132HTR1ADRD2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107344940-B BTK inhibitors and uses thereof 广东东阳光药业有限公司 2020-04-21 CN disclosed