SCHEMBL28396995

SCHEMBL28396995

Nc1nc(N2C(=O)c3ccccc3C2=O)cc(N2C(=O)c3ccccc3C2=O)n1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
CYP3A4 P08684 1/20 0.45
NFKB1 P19838 1/20 0.45
PMP22 Q01453 1/20 0.45
POLB P06746 1/20 0.42
SCN2A Q99250 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HTT P42858 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
HSPA1A P0DMV8 1/20 0.40
PABPC1 P11940 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28397035 0.78 MAP3K5 (0.38) ALDH1A1KDM4EPOLBMEN1KMT2A
SCHEMBL8555373 0.78 ALPL (0.46) ALDH1A1CYP3A4NFKB1PMP22POLB
SCHEMBL5322518 0.78 ALPL (0.44) ALDH1A1CYP3A4NFKB1PMP22POLB
SCHEMBL28400364 0.78 ANPEP (0.35) ALDH1A1KDM4EGAAHSPA1APABPC1
SCHEMBL7250955 0.77 ALDH1A1 (0.49) ALDH1A1KDM4EGAACYP3A4NFKB1
SCHEMBL501398 0.73 KMT2A (0.45) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL11072686 0.73 KMT2A (0.45) ALDH1A1KDM4EGAAPOLBMEN1
SCHEMBL893875 0.73 MEN1 (0.44) ALDH1A1KDM4EGAACYP3A4NFKB1
SCHEMBL8605347 0.72 KMT2A (0.44) ALDH1A1KDM4EGAAMEN1KMT2A
SCHEMBL12617582 0.72 ADORA2A (0.43) ALDH1A1KDM4EGAASCN2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111217839-A 2, 6-disubstituted pyrimidine aromatic anhydride and synthesis method and application thereof 浙江大学 2020-06-02 CN disclosed