SCHEMBL28397978

SCHEMBL28397978

COS(=O)(=O)c1cccc2ccncc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.42
PRKD3 O94806 6/20 0.42
PRKCG P05129 6/20 0.42
PRKCB P05771 6/20 0.42
PRKCA P17252 6/20 0.42
PRKCH P24723 6/20 0.42
PRKCI P41743 6/20 0.42
PRKCE Q02156 6/20 0.42
PRKCQ Q04759 6/20 0.42
PRKCZ Q05513 6/20 0.42
PRKCD Q05655 6/20 0.42
PRKD1 Q15139 6/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2D6 P10635 3/20 0.42
NFKB1 P19838 3/20 0.42
GLA P06280 1/20 0.42
LMNA P02545 2/20 0.41
PMP22 Q01453 1/20 0.41
PRKACA P17612 4/20 0.40
PRKACG P22612 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28399717 0.87 PRKD3 (0.55) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL28394910 0.83 PRKD3 (0.42) TNFPRKD3PRKCGPRKCBPRKCA
SCHEMBL11983469 0.81 TNF (0.46) TNFPRKD3PRKCGPRKCBPRKCA
SCHEMBL29732947 0.79 CA1 (0.57) MEN1KMT2ACA1CA2CA9
SCHEMBL29093707 0.79 CA1 (0.57) MEN1KMT2ACA1CA2CA9
SCHEMBL1002263 0.79 CA1 (0.57) MEN1KMT2ACA1CA2CA9
SCHEMBL3129943 0.78 TNF (0.46) TNFPRKD3PRKCGPRKCBPRKCA
SCHEMBL30002842 0.78 TNF (0.46) TNFPRKD3PRKCGPRKCBPRKCA
SCHEMBL18019196 0.78 CA2 (0.61) TNFPRKD3PRKCGPRKCBPRKCA
SCHEMBL26422606 0.78 TNF (0.46) TNFPRKD3PRKCGPRKCBPRKCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111153856-A Preparation method of fasudil hydrochloride impurity with genotoxicity 湖南增达生物科技有限公司 2020-05-15 CN claimed
CN-111153856-A Preparation method of fasudil hydrochloride impurity with genotoxicity 湖南增达生物科技有限公司 2020-05-15 CN disclosed