SCHEMBL28404175

SCHEMBL28404175

CCOC(=O)c1cc(C)nc(NNC(=O)OC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
RAB9A P51151 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
THRB P10828 1/20 0.42
GAA P10253 3/20 0.42
PDPK1 O15530 1/20 0.42
ALDH1A1 P00352 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30276226 1.00 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL30276208 0.87 LMNA (0.48) CA12CA1CA2CA7CA9
SCHEMBL20937443 0.87 LMNA (0.48) CA12CA1CA2CA7CA9
SCHEMBL12852739 0.77 MEN1 (0.51) CA12CA1CA2CA7CA9
SCHEMBL22840821 0.75 NPC1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL20302320 0.75 LCK (0.46) CA12CA1CA2CA7CA9
SCHEMBL3937264 0.74 LMNA (0.53) CA12CA1CA2CA7CA9
SCHEMBL18773577 0.74 CA12 (0.62) CA12CA1CA2CA7CA9
SCHEMBL1424853 0.73 MEN1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL20937441 0.72 LMNA (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111225915-B Imidazopyridine compounds as PAD inhibitors 朱比兰特埃皮帕德有限公司 2023-03-07 CN disclosed
CN-111225915-A Imidazopyridine compounds as PAD inhibitors 朱比兰特埃皮帕德有限公司 2020-06-02 CN disclosed