SCHEMBL28406191

SCHEMBL28406191

CC#Cc1cccc(C(=O)N(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.49
ERN1 O75460 4/20 0.42
NPSR1 Q6W5P4 1/20 0.40
ACACB O00763 4/20 0.39
MTOR P42345 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PMM2 O15305 1/20 0.39
MPI P34949 1/20 0.39
PHOSPHO1 Q8TCT1 1/20 0.39
KIF11 P52732 1/20 0.39
PIK3CA P42336 1/20 0.39
TRIM24 O15164 1/20 0.39
BRD4 O60885 1/20 0.39
TAF1 P21675 1/20 0.39
SMARCA2 P51531 1/20 0.39
SMARCA4 P51532 1/20 0.39
BRPF1 P55201 1/20 0.39
EP300 Q09472 1/20 0.39
PBRM1 Q86U86 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719359 0.85 PTGDR2 (0.54) PTGDR2ERN1NPSR1ACACBMTOR
SCHEMBL30784948 0.81 GSK3B (0.56) PTGDR2ERN1MEN1KMT2AALDH1A1
SCHEMBL3813604 0.81 GSK3B (0.56) PTGDR2ERN1MEN1KMT2AALDH1A1
SCHEMBL29488328 0.80 CA12 (0.48) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL12724811 0.80 ACACB (0.50) ACACBMEN1KMT2ACREBBPALDH1A1
SCHEMBL27974625 0.80 CA12 (0.48) MEN1KMT2AALDH1A1HPGDSMN1; SMN2
SCHEMBL7406706 0.79 MEN1 (0.55) ERN1MEN1KMT2APMM2MPI
SCHEMBL18946169 0.79 GRM5 (0.55) MEN1KMT2A
SCHEMBL13891405 0.78 ALDH1A1 (0.52) PTGDR2ERN1NPSR1ACACBMTOR
SCHEMBL4672150 0.76 ALDH1A1 (0.51) MEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106496209-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-30 CN disclosed
CN-106496210-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-06-09 CN disclosed
CN-106518856-B Compounds useful as inhibitors of ATR kinase 沃泰克斯药物股份有限公司 2020-04-28 CN disclosed