SCHEMBL28407491

SCHEMBL28407491

Fc1ccc(Nc2ncnc3cc(C4CNCCO4)c(F)cc23)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.57
KDR P35968 2/20 0.52
EPHB4 P54760 2/20 0.52
FBP1 P09467 2/20 0.52
AURKA O14965 1/20 0.52
ERBB2 P04626 1/20 0.52
INSR P06213 1/20 0.52
PDGFRB P09619 1/20 0.52
FLT4 P35916 1/20 0.52
CLK1 P49759 1/20 0.52
TEK Q02763 1/20 0.52
AURKB Q96GD4 1/20 0.52
EPHA2 P29317 3/20 0.51
GRM1 Q13255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28409421 0.84 EGFR (0.61) EGFRERBB2
SCHEMBL28409241 0.83 EPHA2 (0.49) EGFRKDREPHB4EPHA2
SCHEMBL28181389 0.82 EGFR (0.56) EGFRKDREPHB4FBP1AURKA
SCHEMBL28696327 0.78 EPHA2 (0.67) EGFRKDREPHB4FBP1ERBB2
SCHEMBL28403915 0.77 EGFR (0.74) EGFRKDREPHB4FBP1AURKA
SCHEMBL12609963 0.75
SCHEMBL12609961 0.75
SCHEMBL28403896 0.75 EGFR (0.59) EGFRERBB2
SCHEMBL28412441 0.75 EGFR (0.58) EGFRKDREPHB4FBP1AURKA
SCHEMBL27822000 0.74 FBP1 (0.53) EGFRKDREPHB4FBP1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107200715-B Quinazoline derivative and application thereof in preparation of antitumor drugs 陕西师范大学 2020-05-29 CN disclosed