SCHEMBL28409241

SCHEMBL28409241

C/C=C/c1ccc(Nc2ncnc3cc(C4CNCCO4)c(F)cc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EPHA2 P29317 9/20 0.49
EGFR P00533 1/20 0.46
KDR P35968 1/20 0.42
EPHB4 P54760 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28407491 0.83 EGFR (0.57) EPHA2EGFRKDREPHB4
SCHEMBL28181381 0.78 EGFR (0.53) EGFRKDREPHB4
SCHEMBL28181389 0.78 EGFR (0.56) EPHA2EGFRKDREPHB4
SCHEMBL28407194 0.77 EGFR (0.42) EGFR
SCHEMBL28407547 0.77 EGFR (0.49) EPHA2EGFR
SCHEMBL28409415 0.76 EGFR (0.44) EPHA2EGFRKDR
SCHEMBL28182145 0.75 EGFR (0.51) EPHA2EGFRKDREPHB4
SCHEMBL28409421 0.73 EGFR (0.61) EGFR
SCHEMBL28409239 0.73 EGFR (0.63) EPHA2EGFRKDREPHB4
SCHEMBL4890627 0.72 EPHA2 (0.71) EPHA2EGFRKDREPHB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107200715-B Quinazoline derivative and application thereof in preparation of antitumor drugs 陕西师范大学 2020-05-29 CN disclosed