SCHEMBL28407635

SCHEMBL28407635

CC(=CS(C)(=O)=O)CC(NC(=O)OCc1ccccc1)(C(=O)OC(C)C)c1ccc(-c2cnn(C(F)F)c2)cc1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ELANE P08246 4/20 0.33
MGLL Q99685 1/20 0.33
ROCK2 O75116 1/20 0.32
RORC P51449 2/20 0.32
CASP3 P42574 2/20 0.32
EP300 Q09472 3/20 0.31
MMP2 P08253 3/20 0.31
MMP9 P14780 3/20 0.31
MMP3 P08254 2/20 0.31
MMP14 P50281 2/20 0.31
MMP1 P03956 1/20 0.31
MMP7 P09237 1/20 0.31
PTPN1 P18031 2/20 0.31
PTPN2 P17706 1/20 0.31
PTPRB P23467 1/20 0.31
ACP1 P24666 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21149553 1.00 MEN1 (0.33) MEN1KMT2AELANEMGLLROCK2
SCHEMBL28407633 1.00 MEN1 (0.33) MEN1KMT2AELANEMGLLROCK2
SCHEMBL21112221 0.92 MGLL (0.35) MEN1KMT2AELANEMGLLROCK2
SCHEMBL21112222 0.92 MGLL (0.35) MEN1KMT2AELANEMGLLROCK2
SCHEMBL21112223 0.92 MGLL (0.35) MEN1KMT2AELANEMGLLROCK2
SCHEMBL23114939 0.90 MEN1 (0.37) MEN1KMT2AELANEMGLLROCK2
SCHEMBL21149554 0.90 MEN1 (0.37) MEN1KMT2AELANEMGLLROCK2
SCHEMBL29640161 0.89 EP300 (0.35) MEN1KMT2AELANEMGLLROCK2
SCHEMBL21149555 0.89 MEN1 (0.36) MEN1KMT2AELANEMGLLROCK2
SCHEMBL28403733 0.89 MEN1 (0.36) MEN1KMT2AELANEMGLLROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111212832-A 1-benzyl-2-imino-4-phenyl-5-oxoimidazolidine derivatives as HIV protease inhibitors 吉利德科学公司 2020-05-29 CN disclosed