SCHEMBL28414941

SCHEMBL28414941

O=Cc1cc(Br)cc(OCC2CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 2/20 0.42
TLR2 O60603 2/20 0.42
PARP15 Q460N3 5/20 0.38
PARP10 Q53GL7 5/20 0.38
PARP2 Q9UGN5 2/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
KDM1A O60341 1/20 0.36
CHRNB4 P30926 2/20 0.36
CHRNA3 P32297 2/20 0.36
HPGD P15428 2/20 0.34
ALDH1A1 P00352 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4569118 0.92 TLR4 (0.45) TLR4TLR2PARP15PARP10PARP2
SCHEMBL1417220 0.82 CHRNB4 (0.43) PARP15PARP10PARP2CHRNB4CHRNA3
SCHEMBL18003885 0.82 HPGD (0.37) MAOAMAOBCHRNB4CHRNA3HPGD
SCHEMBL20208342 0.81 TLR4 (0.42) TLR4TLR2PARP15PARP10PARP2
SCHEMBL14227724 0.81 TLR4 (0.42) TLR4TLR2PARP15PARP10PARP2
SCHEMBL16247136 0.80 TLR4 (0.50) TLR4TLR2PARP15PARP10PARP2
SCHEMBL18003786 0.79 MAOA (0.34) MAOAMAOBCHRNB4CHRNA3ALDH1A1
SCHEMBL18003300 0.78 HPGD (0.39) MAOAMAOBCHRNB4CHRNA3HPGD
SCHEMBL13746027 0.77 TLR4 (0.39) TLR4TLR2PARP15PARP10PARP2
SCHEMBL27910449 0.77 NR1H4 (0.47) TLR4TLR2PARP15PARP10PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111132961-A Bisaryloxy derivatives as TTX-S blockers 拉夸里亚创药株式会社 2020-05-08 CN disclosed