SCHEMBL28426558

SCHEMBL28426558

CCOC(=O)c1ccc2cccc(I)c2n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
MAPT P10636 1/20 0.50
GAA P10253 1/20 0.45
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MAPK1 P28482 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
TSHR P16473 1/20 0.41
CDC25B P30305 1/20 0.40
FGFR1 P11362 1/20 0.40
FLT1 P17948 1/20 0.40
FGFR3 P22607 1/20 0.40
PDE4A P27815 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17652250 0.84 CYP1A2 (0.63) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL3433286 0.82 CYP1A2 (0.61) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL1209954 0.81 CYP1A2 (0.51) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL2783408 0.81 CYP1A2 (0.59) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL27285116 0.81 CYP1A2 (0.59) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL1478915 0.77 CYP1A2 (1.00) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL13256158 0.76 CYP1A2 (0.77) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL109583 0.76 CYP1A2 (0.82) CYP1A2MAPTGAAKMT2AKDM4E
SCHEMBL28230577 0.76 KDM4E (0.66) KMT2AKDM4ETSHRMEN1
SCHEMBL30253505 0.75 KDM4E (0.64) CYP1A2MAPTGAAKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108314647-B Preparation method of quinoline-2-formic acid and quinoline-2-formic acid derivative 华中科技大学 2020-06-26 CN claimed
CN-108314647-B Preparation method of quinoline-2-formic acid and quinoline-2-formic acid derivative 华中科技大学 2020-06-26 CN disclosed