SCHEMBL28429359

SCHEMBL28429359

CCn1cc(C#N)c2cc(NC(=O)c3ccnc(Cl)c3)ccc21

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 6/20 0.69
CA12 O43570 4/20 0.69
XDH P47989 12/20 0.52
CA2 P00918 1/20 0.50
PFKFB2 O60825 2/20 0.49
PFKFB1 P16118 2/20 0.49
PFKFB3 Q16875 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29940470 1.00 CA9 (0.69) CA9CA12XDHCA2PFKFB2
SCHEMBL29940592 0.92 XDH (0.61) CA9CA12XDH
SCHEMBL28429924 0.92 XDH (0.61) CA9CA12XDH
SCHEMBL28432911 0.89 XDH (0.65) CA9CA12XDH
SCHEMBL29940471 0.89 XDH (0.65) CA9CA12XDH
SCHEMBL29940711 0.89 XDH (0.65) CA9CA12XDH
SCHEMBL28426545 0.89 XDH (0.65) CA9CA12XDH
SCHEMBL29940925 0.88 CA9 (0.55) CA9CA12XDHPFKFB2PFKFB1
SCHEMBL28426663 0.88 CA9 (0.55) CA9CA12XDHPFKFB2PFKFB1
SCHEMBL28896300 0.87 CA9 (0.67) CA9CA12XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111072634-A 1-substituted-3-substituted-5-substituted amide-1H-indole compound and preparation method and application thereof 中国医科大学 2020-04-28 CN claimed
CN-111072634-B 1-substituted-3-substituted-5-substituted amide-1H-indole compound and preparation method and application thereof 中国医科大学 2022-07-22 CN disclosed
CN-111072634-A 1-substituted-3-substituted-5-substituted amide-1H-indole compound and preparation method and application thereof 中国医科大学 2020-04-28 CN disclosed