SCHEMBL28435159

SCHEMBL28435159

CN(C)CCOc1ccc2c(c1)CN(c1nccc(/C=C/c3ccnc(N)c3)n1)C2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.38
ABHD6 Q9BV23 1/20 0.38
TRAP1 Q12931 4/20 0.36
HSP90B1 P14625 3/20 0.36
ROCK2 O75116 3/20 0.35
LCK P06239 2/20 0.34
AURKA O14965 1/20 0.34
JAK2 O60674 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
INSR P06213 1/20 0.34
IGF1R P08069 1/20 0.34
MET P08581 1/20 0.34
KIT P10721 1/20 0.34
FGFR4 P22455 1/20 0.34
CDK2 P24941 1/20 0.34
MAPK1 P28482 1/20 0.34
KDR P35968 1/20 0.34
SYK P43405 1/20 0.34
MAPK8 P45983 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30189613 0.93 MGLL (0.35) MGLLABHD6TRAP1HSP90B1ROCK2
SCHEMBL22229569 0.93 MGLL (0.35) MGLLABHD6TRAP1HSP90B1ROCK2
SCHEMBL28451045 0.86 ROCK2 (0.48) ROCK2ROCK1HSP90AA1NOS1NOS2
SCHEMBL22229621 0.82 ROCK2 (0.39) MGLLABHD6TRAP1HSP90B1ROCK2
SCHEMBL30189612 0.82 ROCK2 (0.39) MGLLABHD6TRAP1HSP90B1ROCK2
SCHEMBL28443783 0.78 KDM4E (0.42) ROCK2ROCK1KDM4E
SCHEMBL28897461 0.78 GRM4 (0.34) ROCK2ROCK1KDM4EHSP90AA1
SCHEMBL28437048 0.78 GRM4 (0.44) ROCK2ROCK1KDM4EHRH3ADORA2A
SCHEMBL22229650 0.78 ROCK2 (0.43) ROCK2ROCK1NOS1NOS2
SCHEMBL30189463 0.78 ROCK2 (0.43) ROCK2ROCK1NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111406051-A Vinylheterocycles as RHO-associated coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2020-07-10 CN claimed
CN-111406051-A Vinylheterocycles as RHO-associated coiled coil kinase (ROCK) inhibitors 安吉昂生物医药公司 2020-07-10 CN disclosed