SCHEMBL28435645

SCHEMBL28435645

Cc1nccn1-c1nc(Cl)c(F)c(Cl)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2E1 P05181 1/20 0.39
CYP2A6 P11509 1/20 0.39
PIK3CA P42336 3/20 0.36
MTOR P42345 3/20 0.36
TUBB4A P04350 2/20 0.35
TUBB P07437 2/20 0.35
TUBA3C P0DPH7 2/20 0.35
TUBA1B P68363 2/20 0.35
TUBA4A P68366 2/20 0.35
TUBB4B P68371 2/20 0.35
TUBB3 Q13509 2/20 0.35
TUBB2A Q13885 2/20 0.35
TUBB8 Q3ZCM7 2/20 0.35
TUBA3E Q6PEY2 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026494 0.80 CYP3A4 (0.48) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL12918510 0.73 CYP3A4 (0.43) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL27961165 0.72 TSHR (0.49) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL20154101 0.70 PIK3CA (0.53) ALDH1A1KDM4EPIK3CAMTORLMNA
SCHEMBL31205699 0.68 RPS6KA5 (0.52) ALDH1A1KMT2ACYP3A4CYP2E1CYP2A6
SCHEMBL28728263 0.67 CYP3A4 (0.48) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL2666367 0.67 CYP3A4 (0.44) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL19764720 0.66 MAOA (0.53) ALDH1A1KDM4EMEN1HPGDKMT2A
SCHEMBL12342913 0.66 CYP3A4 (0.47) ALDH1A1KDM4ECYP3A4CYP2E1CYP2A6
SCHEMBL19211560 0.64 KDR (0.52) ALDH1A1CYP3A4CYP2E1CYP2A6TUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423417-B Substituted reverse pyrimidine Bmi-1 inhibitors PTC医疗公司 2022-11-15 CN disclosed
CN-111423417-A Substituted reverse pyrimidine Bmi-1 inhibitors PTC医疗公司 2020-07-17 CN disclosed