SCHEMBL28435874

SCHEMBL28435874

CCOC(=O)CC(=O)C1C[C@H](c2c(F)ccc(Br)c2F)CN1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
KDM4E B2RXH2 2/20 0.34
TSHR P16473 1/20 0.34
CHRM1 P11229 1/20 0.31
HCRTR2 O43614 3/20 0.30
NLRP3 Q96P20 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21052749 1.00 ALDH1A1 (0.34) ALDH1A1KDM4ETSHRCHRM1HCRTR2
SCHEMBL28431241 1.00 ALDH1A1 (0.34) ALDH1A1KDM4ETSHRCHRM1HCRTR2
SCHEMBL23455095 0.92 HCRTR2 (0.36) ALDH1A1CHRM1HCRTR2NLRP3
SCHEMBL21052694 0.92 HCRTR2 (0.36) ALDH1A1CHRM1HCRTR2NLRP3
SCHEMBL21054669 0.88 ALDH1A1 (0.34) ALDH1A1KDM4ETSHR
SCHEMBL21053552 0.88 ALDH1A1 (0.34) ALDH1A1KDM4ETSHR
SCHEMBL23455038 0.88 CYP1A2 (0.35) IDO1
SCHEMBL23454789 0.88 CYP1A2 (0.35) IDO1
SCHEMBL23455039 0.88 CYP1A2 (0.35) IDO1
SCHEMBL23454788 0.88 CYP1A2 (0.35) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111479812-A dopamine-B-hydroxylase inhibitors 巴尔-波特拉及康邦亚股份有限公司 2020-07-31 CN disclosed