SCHEMBL21054669

SCHEMBL21054669

CCOC(=O)CC(=O)C1CC(c2c(F)ccc(Cl)c2F)CN1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 2/20 0.34
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 6/20 0.33
MEN1 O00255 4/20 0.33
ATM Q13315 2/20 0.33
MGLL Q99685 2/20 0.33
ALOX15 P16050 1/20 0.33
S1PR1 P21453 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HPGD P15428 1/20 0.31
GAA P10253 2/20 0.31
PPOX P50336 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21053552 1.00 ALDH1A1 (0.34) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL23455095 0.92 HCRTR2 (0.36) ALDH1A1GAA
SCHEMBL21052694 0.92 HCRTR2 (0.36) ALDH1A1GAA
SCHEMBL28431241 0.88 ALDH1A1 (0.34) ALDH1A1KDM4ETSHR
SCHEMBL21052749 0.88 ALDH1A1 (0.34) ALDH1A1KDM4ETSHR
SCHEMBL28435874 0.88 ALDH1A1 (0.34) ALDH1A1KDM4ETSHR
SCHEMBL29891871 0.88 USP30 (0.37) ALDH1A1SMN1; SMN2POLBKMT2AMEN1
SCHEMBL29891600 0.88 USP30 (0.37) ALDH1A1SMN1; SMN2POLBKMT2AMEN1
SCHEMBL21053205 0.86 NLRP3 (0.40) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL28434356 0.86 NLRP3 (0.40) ALDH1A1KDM4ETSHRTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3720856-A1 DOPAMINE-& X392;-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2020-10-14 EP disclosed
WO-2019112457-A1 DOPAMINE-Β-HYDROXYLASE INHIBITORS BIAL - PORTELA & Cª, S.A. (PT) 2019-06-13 WO disclosed