SCHEMBL28439760

SCHEMBL28439760

O=C(CCl)n1ccc2cc(O)cnc21

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 10/20 0.38
SLC22A6 Q4U2R8 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
FGFR1 P11362 2/20 0.37
FGFR4 P22455 2/20 0.37
ENPP3 O14638 3/20 0.36
ENPP1 P22413 2/20 0.36
PARP1 P09874 1/20 0.36
GSK3B P49841 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24450111 0.72 PIK3CA (0.40) SLC22A12ENPP3ENPP1PARP1
SCHEMBL19708331 0.68 MAP4K4 (0.34)
SCHEMBL1269052 0.68 APP (0.43)
SCHEMBL28055645 0.68 GLO1 (0.37)
SCHEMBL17253109 0.65 DGAT1 (0.37) FGFR1FGFR4
SCHEMBL10837613 0.64 NOTUM (0.59)
SCHEMBL23327801 0.64 SLC22A12 (0.41) SLC22A12SLC22A6ENPP3ENPP1PARP1
SCHEMBL28659326 0.64 PARP1 (0.41) SLC22A12SLC22A6ABCG2FGFR1FGFR4
SCHEMBL21958555 0.64 DGAT1 (0.38)
SCHEMBL9789003 0.62 TFPI2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108456207-B Amide derivative and application thereof in cardiovascular and cerebrovascular aspects 浙江药苑生物科技有限公司 2020-11-20 CN disclosed
CN-108383838-B Amide derivative and application thereof in hypertension, hyperlipidemia and atherosclerosis 浙江药苑生物科技有限公司 2020-08-28 CN disclosed
CN-108218865-B Amide derivative and application thereof in cardiovascular and cerebrovascular aspects 济南市儿童医院 2020-06-26 CN disclosed