SCHEMBL2844248

SCHEMBL2844248

O=C(Cc1ccc(C(c2ccc(F)cc2)N2CCCCC2)c(-c2ccc(C(F)(F)F)cc2)c1)N1C(=O)OC[C@H]1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.47
PSEN1 P49768 2/20 0.47
PSEN2 P49810 2/20 0.47
APH1B Q8WW43 2/20 0.47
NCSTN Q92542 2/20 0.47
APH1A Q96BI3 2/20 0.47
PSENEN Q9NZ42 2/20 0.47
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
CACNA2D1 P54289 2/20 0.35
CACNA1B Q00975 2/20 0.35
CACNB1 Q02641 2/20 0.35
CACNA1C Q13936 2/20 0.35
CACNA1A O00555 1/20 0.35
P4HB P07237 6/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
TACR1 P25103 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2845339 0.86 KCNH2 (0.49) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL2844020 0.85 KCNH2 (0.47) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL2850124 0.81 KCNH2 (0.58) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL2847936 0.76 KCNH2 (0.55) KCNH2PSEN1PSEN2APH1BNCSTN
SCHEMBL5767504 0.74 TACR1 (0.44) TACR1
SCHEMBL5765764 0.74 TACR1 (0.44) TACR1
SCHEMBL2559137 0.74 CACNA1G (0.43) CNR1
SCHEMBL16680346 0.74 CACNA1G (0.43) CNR1
SCHEMBL2559140 0.74 CACNA1G (0.43) CNR1
SCHEMBL2878111 0.73 KCNH2 (0.62) KCNH2PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010138901-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS, DERIVATIVES THEREOF, AND RELATED METHODS OF USE BIOGEN IDEC MA INC (US) 2010-12-02 WO disclosed