SCHEMBL16680346

SCHEMBL16680346

O=C(Cc1ccc(F)cc1)N1C(=O)OC[C@H]1Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.43
NAAA Q02083 2/20 0.42
FAAH O00519 4/20 0.41
CNR1 P21554 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
IL6ST P40189 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
ALOX12 P18054 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
CASP3 P42574 1/20 0.40
CASP7 P55210 1/20 0.40
MC4R P32245 2/20 0.40
MC3R P41968 2/20 0.40
MC1R Q01726 2/20 0.40
TACR3 P29371 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2559140 1.00 CACNA1G (0.43) CACNA1GNAAAFAAHCNR1SIGMAR1
SCHEMBL2559137 1.00 CACNA1G (0.43) CACNA1GNAAAFAAHCNR1SIGMAR1
SCHEMBL1915646 0.92 NAAA (0.47) NAAAFAAHIL6STALDH1A1MC4R
SCHEMBL7346791 0.92 NAAA (0.47) NAAAFAAHIL6STALDH1A1MC4R
SCHEMBL1915643 0.92 NAAA (0.47) NAAAFAAHIL6STALDH1A1MC4R
SCHEMBL23866771 0.88 NAAA (0.51) NAAAFAAHIL6STPKMALDH1A1
SCHEMBL23902846 0.88 NAAA (0.51) NAAAFAAHIL6STPKMALDH1A1
SCHEMBL23860312 0.88 NAAA (0.42) NAAAFAAHSIGMAR1IL6STMC4R
SCHEMBL21871072 0.88 NAAA (0.42) NAAAFAAHSIGMAR1IL6STMC4R
SCHEMBL23522276 0.88 NAAA (0.51) NAAAFAAHIL6STPKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9452990-B2 Complement pathway modulators and uses thereof NOVARTIS AG (CH) 2016-09-27 US disclosed
EP-2864322-B1 COMPLEMENT PATHWAY MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2016-04-27 EP disclosed
US-20150126492-A1 Complement Pathway Modulators and Uses Thereof NOVARTIS AG (CH) 2015-05-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150126492-A1 Complement Pathway Modulators and Uses Thereof CFB, CFH, TFPI CACNA1G 4528/4885NAAA 4222/4885FAAH 1826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.