SCHEMBL2844330

SCHEMBL2844330

C/C(=N\O)c1ccc(C(C)C(=O)O)cc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 15/20 0.62
AKR1C2 P52895 15/20 0.62
PTGS1 P23219 4/20 0.48
PTGS2 P35354 3/20 0.48
KCNH2 Q12809 2/20 0.48
PSEN1 P49768 2/20 0.48
PSEN2 P49810 2/20 0.48
APH1B Q8WW43 2/20 0.48
NCSTN Q92542 2/20 0.48
APH1A Q96BI3 2/20 0.48
PSENEN Q9NZ42 2/20 0.48
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
APP P05067 1/20 0.43
CYP3A4 P08684 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
FABP2 P12104 1/20 0.43
TSHR P16473 1/20 0.43
AKR1C4 P17516 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597658 0.79 AKR1C3 (0.74) AKR1C3AKR1C2PTGS1PTGS2KCNH2
SCHEMBL1372793 0.77 AKR1C3 (1.00) AKR1C3AKR1C2PTGS1PTGS2PSEN1
SCHEMBL2848165 0.77 AKR1C3 (0.67) AKR1C3AKR1C2PTGS1PTGS2KCNH2
SCHEMBL2844333 0.76 AKR1C3 (0.59) AKR1C3AKR1C2PTGS1PTGS2KCNH2
SCHEMBL23354256 0.74 AKR1C3 (0.52) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL1797371 0.74 AKR1C3 (0.65) AKR1C3AKR1C2PTGS1PTGS2PSEN1
SCHEMBL2848167 0.74 AKR1C3 (0.66) AKR1C3AKR1C2PTGS1PTGS2KCNH2
SCHEMBL7805874 0.72 PSEN1 (0.49) AKR1C3AKR1C2PSEN1PSEN2APH1B
SCHEMBL6270587 0.71 AKR1C3 (0.63) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL4596111 0.70 AKR1C3 (0.61) AKR1C3AKR1C2PTGS1PTGS2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010138901-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS, DERIVATIVES THEREOF, AND RELATED METHODS OF USE BIOGEN IDEC MA INC (US) 2010-12-02 WO disclosed