SCHEMBL28445463

SCHEMBL28445463

CCOC(=O)CCc1nc2ccc(Br)cc2nc1Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
HSD17B10 Q99714 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
EGFR P00533 1/20 0.39
MAPT P10636 2/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NAMPT P43490 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SCN9A Q15858 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28451603 1.00 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28443100 0.94 KDM4E (0.44) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28449263 0.90 KDM4E (0.52) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28443132 0.88 MAPT (0.46) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28898030 0.88 HDAC6 (0.51) KDM4EL3MBTL1HDAC6MCL1
SCHEMBL28447953 0.88 HDAC6 (0.51) KDM4EL3MBTL1HDAC6MCL1
SCHEMBL28449191 0.85 EGFR (0.43) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28452127 0.85 KMT2A (0.40) ALDH1A1KDM4ELMNAHSD17B10EGFR
SCHEMBL28443055 0.83 KDM4E (0.54) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1
SCHEMBL28445422 0.82 KDM4E (0.44) ALDH1A1KDM4ELMNAHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108997230-B Quinoxaline derivative with matrix metalloproteinase inhibitory activity, preparation method and application thereof 山东大学 2020-08-04 CN claimed
CN-108997230-B Quinoxaline derivative with matrix metalloproteinase inhibitory activity, preparation method and application thereof 山东大学 2020-08-04 CN disclosed